SCHEMBL8515228

SCHEMBL8515228

CC1(C)CN=C(c2ccc(Cl)cc2N)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
TSHR P16473 3/20 0.40
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.35
CNR1 P21554 3/20 0.34
CNR2 P34972 3/20 0.34
ABL1 P00519 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9607169 0.89 IDO1 (0.39) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL9607171 0.78 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2TDP1GAAKMT2A
SCHEMBL9607464 0.77 CNR2 (0.32) CNR2
SCHEMBL9607342 0.77 CNR2 (0.32) CNR2
SCHEMBL9607484 0.75 CNR2 (0.34) CNR2
SCHEMBL27185985 0.68 ALDH1A1 (0.65) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL30839752 0.68 ALDH1A1 (0.65) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL30839712 0.68 ALDH1A1 (0.65) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL19002042 0.67 CYP3A4 (0.40) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL23580463 0.66 CNR2 (0.34) ALDH1A1SMN1; SMN2CNR2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed