SCHEMBL8517181

SCHEMBL8517181

C=CCOc1ccc(-c2ccc(C#CC(C)O)nc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.45
ACACB O00763 4/20 0.41
MCHR1 Q99705 8/20 0.39
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
CHRM1 P11229 2/20 0.35
HTR2A P28223 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517151 0.85 CYP2D6 (0.43) CYP2D6ACACBMCHR1ADRB2ADRB1
SCHEMBL8517707 0.84 CYP2D6 (0.51) CYP2D6ACACBMCHR1ADRB2ADRB1
SCHEMBL8517135 0.83 CYP2D6 (0.43) CYP2D6ACACBMCHR1ADRB2ADRB1
SCHEMBL8518327 0.82 ACACB (0.40) CYP2D6ACACBMCHR1KDM4EALDH1A1
SCHEMBL8517335 0.79 CYP2D6 (0.44) CYP2D6ACACBMCHR1ADRB2ADRB1
SCHEMBL7554101 0.77 ACACB (0.36) CYP2D6ACACBMCHR1KDM4EALDH1A1
SCHEMBL8517796 0.75 CYP2D6 (0.43) CYP2D6ACACBADRB2ADRB1ADRB3
SCHEMBL8517137 0.73 CYP2D6 (0.48) CYP2D6ADRB2ADRB1ADRB3ALDH1A1
SCHEMBL10581510 0.72 CYP2D6 (0.52) CYP2D6ADRB2ADRB1ADRB3KDM4E
SCHEMBL472165 0.71 CA12 (0.57) CYP2D6KDM4EALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed