SCHEMBL8517137

SCHEMBL8517137

C=CCOc1ccc2cc(C#CC(C)O)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.48
CA12 O43570 5/20 0.43
CA1 P00915 5/20 0.43
CA9 Q16790 5/20 0.43
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADRB2 P07550 2/20 0.39
ADRB1 P08588 2/20 0.39
ADRB3 P13945 2/20 0.39
SRC P12931 2/20 0.38
ABL1 P00519 1/20 0.38
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517707 0.85 CYP2D6 (0.51) CYP2D6CA12CA1CA9NPC1
SCHEMBL8679613 0.78 ABCB11 (0.45) CYP2D6MEN1LMNAMAPTKMT2A
SCHEMBL8517544 0.78 ALDH1A1 (0.41) NPC1TP53RAB9AMEN1LMNA
SCHEMBL8517269 0.78 CYP2D6 (0.35) CYP2D6LMNASMN1; SMN2ADRB2ADRB1
SCHEMBL8517666 0.78 CYP2D6 (0.40) CYP2D6CA12CA1CA9MEN1
SCHEMBL8375925 0.77 NR5A1 (0.48) NPC1TP53RAB9ALMNAMAPT
SCHEMBL8517335 0.77 CYP2D6 (0.44) CYP2D6CA12CA1CA9NPC1
SCHEMBL3825460 0.75 CA12 (0.64) CA12CA1CA9NPC1TP53
SCHEMBL8597099 0.75 CA12 (0.38) CYP2D6CA12CA1CA9NPC1
SCHEMBL8517796 0.75 CYP2D6 (0.43) CYP2D6CA12CA1CA9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed