SCHEMBL8517335

SCHEMBL8517335

C=CCOc1ccc(-c2ccc(C#CC(C)O)cn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
HPGD P15428 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 1/20 0.40
MCHR1 Q99705 1/20 0.38
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 2/20 0.34
NPC1 O15118 2/20 0.34
TP53 P04637 1/20 0.34
ACACB O00763 2/20 0.34
GRM5 P41594 1/20 0.34
ABL1 P00519 1/20 0.34
SRC P12931 1/20 0.34
MGAM O43451 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517707 0.86 CYP2D6 (0.51) CYP2D6ALDH1A1KDM4EHPGDMCHR1
SCHEMBL8517151 0.84 CYP2D6 (0.43) CYP2D6ALDH1A1KDM4EMCHR1ADRB2
SCHEMBL8517876 0.84 RAB9A (0.35) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL8517135 0.82 CYP2D6 (0.43) CYP2D6ALDH1A1KDM4EL3MBTL1MCHR1
SCHEMBL9286998 0.80 KDM4E (0.37) CYP2D6ALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL8517181 0.79 CYP2D6 (0.45) CYP2D6ALDH1A1KDM4EMCHR1ADRB2
SCHEMBL7554909 0.78 ALDH1A1 (0.38) CYP2D6ALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL8517137 0.77 CYP2D6 (0.48) CYP2D6ALDH1A1ADRB2ADRB1ADRB3
SCHEMBL7557875 0.77 KDM4E (0.38) CYP2D6ALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL9286994 0.77 KDM4E (0.35) CYP2D6ALDH1A1KDM4EHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed