SCHEMBL8517869

SCHEMBL8517869

CC(C)(C)OC(=O)NC(CCCNCCC#N)C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.52
CTSK P43235 12/20 0.52
CTSL P07711 2/20 0.45
CTSB P07858 2/20 0.45
P2RY2 P41231 1/20 0.42
JAK3 P52333 1/20 0.41
BTK Q06187 1/20 0.41
ATM Q13315 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20817325 0.85 CTSS (0.56) CTSSCTSKCTSLCTSB
SCHEMBL20817323 0.85 CTSS (0.56) CTSSCTSKCTSLCTSB
SCHEMBL7787845 0.83 CTSS (0.52) CTSSCTSKCTSLCTSBP2RY2
SCHEMBL3957707 0.83 MEN1 (0.52) CTSSCTSKP2RY2JAK3BTK
SCHEMBL27923119 0.80 CTSS (0.59) CTSSCTSKCTSLCTSB
SCHEMBL7945007 0.79 TDP1 (0.46) CTSSCTSKP2RY2JAK3BTK
SCHEMBL7787879 0.79 CTSK (0.51) CTSSCTSKCTSLCTSBP2RY2
SCHEMBL19944850 0.78 CTSS (0.55) CTSSCTSKCTSLCTSB
SCHEMBL1603288 0.78 CTSS (0.63) CTSSCTSKCTSLCTSB
SCHEMBL16095226 0.78 CTSS (0.63) CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001824-A Butyryl-tyrosinyl spermine, analogs thereof and methods of preparing and using same THE TRUSTEES OF COLUMBIA UNIVERSITY (US) 1999-12-14 US disclosed
WO-1996022962-A9 BUTYRYL-TYROSINYL SPERMINE, ANALOGS THEREOF AND METHODS OF PREPARING AND USING SAME 1996-10-03 WO disclosed
WO-1996022962-A1 BUTYRYL-TYROSINYL SPERMINE, ANALOGS THEREOF AND METHODS OF PREPARING AND USING SAME THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-08-01 WO disclosed