SCHEMBL8518740

SCHEMBL8518740

CCCCCCCCC=CCCCCCCCC(=O)NC(=O)C(C)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASAH2 Q9NR71 1/20 0.57
HRH3 Q9Y5N1 1/20 0.54
FAAH O00519 4/20 0.54
DEGS1 O15121 1/20 0.53
TERT O14746 3/20 0.53
CYP1A2 P05177 2/20 0.53
MAPT P10636 2/20 0.53
CYP2C19 P33261 2/20 0.53
BLM P54132 2/20 0.53
HSD17B10 Q99714 2/20 0.53
FABP4 P15090 2/20 0.53
PTPN1 P18031 2/20 0.53
PPARG P37231 2/20 0.53
KMT2A Q03164 2/20 0.53
PPARD Q03181 2/20 0.53
PPARA Q07869 2/20 0.53
GMNN O75496 1/20 0.53
USP2 O75604 1/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518730 1.00 ASAH2 (0.57) ASAH2HRH3FAAHDEGS1TERT
SCHEMBL22471671 0.85 FAAH (0.55) ASAH2HRH3FAAHDEGS1TERT
SCHEMBL4815645 0.85 FAAH (0.55) ASAH2HRH3FAAHDEGS1TERT
SCHEMBL9517250 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL10488884 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL424098 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL8150267 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL422846 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL5077835 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT
SCHEMBL2703278 0.85 TERT (0.66) HRH3FAAHTERTCYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5910490-A INHIBITION OF MEMBRANE RECEPTORS FOR ELASTIN WHICH ARE INVOLVED IN DEGRADATION OF FIBROUS STROMA OF THE CONNECTIVE TISSUE ROC. S.A. (FR) 1999-06-08 US disclosed
EP-0714284-A1 USE OF OLIGOSACCHARIDES FOR THE PREVENTION AND TREATMENT OF TISSUE AGEING ROC S.A. (FR) 1996-06-05 EP disclosed
WO-1995005155-A1 USE OF OLIGOSACCHARIDES FOR THE PREVENTION AND TREATMENT OF TISSUE AGEING ROC S.A. (FR) 1995-02-23 WO disclosed
US-4512903-A Lubricant compositions containing amides of hydroxy-substituted aliphatic acids and fatty amines TEXACO INC. (US) 1985-04-23 US disclosed