SCHEMBL852083

SCHEMBL852083

COC(=O)c1ccccc1C=CC#N.COC(=O)c1ccccc1C=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
LMNA P02545 2/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 2/20 0.42
CFTR P13569 1/20 0.41
POLB P06746 2/20 0.41
ATM Q13315 1/20 0.41
RAB9A P51151 1/20 0.40
PIM1 P11309 1/20 0.39
PIM3 Q86V86 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA5A P35218 1/20 0.38
CA9 Q16790 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 1/20 0.38
SLC6A3 Q01959 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL852020 0.94 BACE1 (0.51) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL852019 0.94 BACE1 (0.51) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL30635255 0.84 LMNA (0.57) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL121356 0.84 LMNA (0.57) BACE1LMNATSHRALDH1A1KDM4E
Benzene SCHEMBL28217563 0.83 TSHR (0.55) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL7659268 0.80 BACE1 (0.52) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL69552 0.79 BACE1 (0.60) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL69553 0.79 BACE1 (0.60) BACE1LMNATSHRALDH1A1KDM4E
SCHEMBL852816 0.75 KDM4E (0.46) LMNAALDH1A1KDM4EHSD17B10ATM
SCHEMBL852815 0.75 KDM4E (0.46) LMNAALDH1A1KDM4EHSD17B10ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432783-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2012-03-28 EP disclosed
WO-2010135560-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-11-25 WO disclosed