SCHEMBL8520839

SCHEMBL8520839

O=C(c1cccc2ccccc12)N1CCN(C(Cc2ccc(C(F)(F)F)cc2)c2cnc[nH]2)CC1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
FNTA P49354 11/20 0.45
FNTB P49356 11/20 0.45
TACR1 P25103 2/20 0.43
DRD4 P21917 1/20 0.41
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8152940 0.89 FNTA (0.48) ALDH1A1LMNAFNTAFNTB
SCHEMBL8153147 0.87 FNTA (0.47) ALDH1A1LMNAFNTAFNTB
SCHEMBL8541422 0.86 ALDH1A1 (0.53) ALDH1A1LMNAFNTAFNTB
SCHEMBL7483971 0.86 FNTA (0.47) ALDH1A1LMNAFNTAFNTB
Hydrochloric Acid SCHEMBL7482278 0.85 FNTA (0.47) ALDH1A1LMNAFNTAFNTB
SCHEMBL3499735 0.84 FNTA (0.58) ALDH1A1LMNAFNTAFNTBTACR1
Trifluoroacetic Acid SCHEMBL8452331 0.82 FNTA (0.56) FNTAFNTBTACR1DRD4
SCHEMBL8522108 0.81 FNTA (0.49) ALDH1A1LMNAFNTAFNTB
SCHEMBL7483881 0.76 FNTA (0.38) FNTAFNTBDRD4
Hydrochloric Acid SCHEMBL7748868 0.76 FNTA (0.38) FNTAFNTBDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0952842-A2 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 1999-11-03 EP disclosed
WO-1997038664-A2 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1997-10-23 WO disclosed