SCHEMBL8522230

SCHEMBL8522230

Cc1c(C)c2c(c(C)c1OCc1ccccc1)[C@H](CN1CCC[C@H]1COc1ccc(C=O)cc1)C(C)(C)O2

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.39
MCHR1 Q99705 2/20 0.39
FAAH O00519 6/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNA5 P30532 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
KDM4E B2RXH2 1/20 0.33
SPHK2 Q9NRA0 2/20 0.32
SPHK1 Q9NYA1 2/20 0.32
FFAR1 O14842 1/20 0.32
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961833 0.92 FAAH (0.41) KCNH2MCHR1FAAHCHRNB2SPHK2
SCHEMBL6963235 0.90 FAAH (0.40) KCNH2MCHR1FAAHCHRNB2CHRNA5
SCHEMBL6963231 0.90 FAAH (0.40) KCNH2MCHR1FAAHCHRNB2CHRNA5
SCHEMBL6967496 0.89 HPGD (0.47)
SCHEMBL6969419 0.89 HPGD (0.47)
SCHEMBL6970975 0.89 HPGD (0.47)
SCHEMBL6976242 0.89 FAAH (0.46) KCNH2MCHR1FAAHCHRNB2CHRNA5
SCHEMBL6976244 0.89 FAAH (0.46) KCNH2MCHR1FAAHCHRNB2CHRNA5
Hydrochloric Acid SCHEMBL6958761 0.88 HPGD (0.47)
Maleic Acid SCHEMBL6974160 0.85 HPGD (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894089-A1 NOVEL HETEROCYCLIC COMPOUNDS HAVING ANTIDIABETIC, HYPOLIPIDAEMIC, ANTIHYPERTENSIVE PROPERTIES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-02-03 EP disclosed
WO-1997041121-A1 NOVEL HETEROCYCLIC COMPOUNDS HAVING ANTIDIABETIC, HYPOLIPIDAEMIC, ANTIHYPERTENSIVE PROPERTIES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1997-11-06 WO disclosed