SCHEMBL852255

SCHEMBL852255

O=C1Nc2ccccc2N(C2CCN(C3(C(=O)OCc4ccccc4)CCCCCCC3)CC2)C1Cl

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 4/20 0.40
GAA P10253 2/20 0.40
NPC1 O15118 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL854436 0.81 OPRM1 (0.40) FKBP1AGAANPC1MAPK1RAB9A
SCHEMBL16714152 0.75 OPRM1 (0.38) FKBP1AGAANPC1MAPK1RAB9A
SCHEMBL855707 0.73 OGFRL1 (0.39) FKBP1AGAANPC1MAPK1RAB9A
SCHEMBL551433 0.73 DDB1 (0.48) FKBP1ADDB1CRBN
SCHEMBL550752 0.72 OPRM1 (0.53) OPRM1OPRL1
SCHEMBL25554839 0.71 TSHR (0.49)
SCHEMBL13221719 0.71 OGFRL1 (0.52) OPRM1OPRL1
SCHEMBL551499 0.68 KDM4E (0.44) FKBP1AGAAKDM4EMAPT
SCHEMBL3724255 0.67 DDB1 (0.48) DDB1CRBN
SCHEMBL550300 0.66 CTSL (0.42) FKBP1ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433937-A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof Purdue Pharma LP (US) 2012-03-28 EP disclosed