SCHEMBL852318

SCHEMBL852318

CCCCCCCCCCCCCCCC(=O)N1CCC(O)C1(C(=O)O)C(=O)CCCCCCCCCCCCCCC

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GNAI3 P08754 9/20 0.46
GNAI1 P63096 9/20 0.46
GNAO1 P09471 8/20 0.46
L3MBTL1 Q9Y468 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NAAA Q02083 2/20 0.37
FAAH O00519 1/20 0.37
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
GPR84 Q9NQS5 1/20 0.35
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14166247 0.99 GNAI3 (0.45) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL10494121 0.80 GNAI3 (0.43) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL10616841 0.75 L3MBTL1 (0.42) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL5314499 0.71 GNAI3 (0.38) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL249960 0.71 GNAI3 (0.38) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL28757738 0.71 GNAI3 (0.38) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL5314497 0.71 GNAI3 (0.38) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL28384679 0.70 L3MBTL1 (0.46) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL28142318 0.70 L3MBTL1 (0.46) GNAI3GNAI1GNAO1L3MBTL1MEN1
SCHEMBL14166250 0.70 GNAI3 (0.37) GNAI3GNAI1GNAO1L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 219 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3212688-B1 THERMOPLASTIC POLYURETHANE FILM FOR DELIVERY OF ACTIVE AGENTS TO SKIN SURFACES LUBRIZOL ADVANCED MAT INC (US) 2022-04-13 EP claimed
US-11241373-B2 Cosmetic composition of dispersion formulation comprising spherical particle AMOREPACIFIC CORPORATION (KR) 2022-02-08 US claimed
US-20200214954-A1 COSMETIC COMPOSITION OF DISPERSION FORMULATION COMPRISING SPHERICAL PARTICLE AMOREPACIFIC CORPORATION (KR) 2020-07-09 US claimed
EP-3662881-A2 DISPERSION FORMULATION OF COSMETIC COMPOSITION COMPRISING SPHERICAL PARTICLES Amorepacific Corporation (KR) 2020-06-10 EP claimed
EP-3271012-B1 DEVICES FOR PROVIDING SKIN CARE USING PHOTOTHERAPY INDERM (FR) 2019-06-19 EP claimed
US-20180071547-A1 Methods of Providing Skin Care Using Phototherapy INDERM (FR) 2018-03-15 US claimed
EP-3271012-A1 METHODS OF PROVIDING SKIN CARE USING PHOTOTHERAPY Inderm (FR) 2018-01-24 EP claimed
WO-2016146778-A1 METHODS OF PROVIDING SKIN CARE USING PHOTOTHERAPY INDERM (FR) 2016-09-22 WO claimed
EP-2575861-B1 A NOVEL SYNERGISTIC PHARMACEUTICAL COMPOSITION FOR TOPICAL APPLICATIONS BHARAT BIOTECH INT LTD (IN) 2015-11-04 EP claimed
EP-2445477-B1 COSMETIC COMPOSITION MADE FROM ION-EXCHANGE RESINS FILLED WITH LIPOAMINOACIDS SEPPIC SA (FR) 2015-02-11 EP claimed
WO-2006053688-A1 COSMETIC AND DERMATOLOGICAL PREPARATIONS FOR THE TREATMENT OF MATURE SKIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2006-05-26 WO claimed
WO-2006042627-A2 COSMETIC AND DERMATOLOGICAL COMPOSITIONS CONTAINING ACTIVE SUBSTANCES FOR IMPROVING SENSORY PERCEPTION HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2006-04-27 WO claimed
EP-1640041-A2 Cosmetic and dermatological composition for the treatment of aging or photodamaged skin Henkel Kommanditgesellschaft auf Aktien (DE) 2006-03-29 EP claimed
WO-2006018198-A1 COSMETIC AND DERMATOLOGICAL COMPOSITIONS COMPRISING (2-HYDROXYETHYL)UREA HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2006-02-23 WO claimed
US-RE38441-E1 Solvent-based non-drying lipstick MAYBELLINE, INC. 2004-02-24 US claimed
EP-0874640-B1 CYCLOSPORIN FORMULATION IVAX CR A S (CZ) 2003-07-23 EP claimed
US-5690918-A WAX BASE MAYBELLINE, INC. (US) 1997-11-25 US claimed
EP-0642339-A1 DIPALMITOYLHYDROXYPROLINE AND OLEOYLMETHIONINE CONTAINING COMPOSITION Morelle, J.V. (FR) 1995-03-15 EP claimed
WO-1993023028-A1 DIPALMITOYLHYDROXYPROLINE AND OLEOYLMETHIONINE CONTAINING COMPOSITION MORELLE JEAN (FR) 1993-11-25 WO claimed
EP-0424282-B1 SUN TANNING COSMETIC PREPARATION ERPHAR Société d'Etudes et de Recherches Pharmaceutiques et Cosmétiques (FR) 1993-03-03 EP claimed