SCHEMBL8523787

SCHEMBL8523787

Cc1nc2c(O)n(-c3ccc(Cl)cc3)nc2c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 2/20 0.52
CA9 Q16790 1/20 0.44
GRM1 Q13255 2/20 0.41
GRM5 P41594 1/20 0.41
LMNA P02545 1/20 0.40
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ESR2 Q92731 1/20 0.38
GABRA1 P14867 2/20 0.37
GABRA2 P47869 2/20 0.37
HTT P42858 2/20 0.37
AURKA O14965 1/20 0.37
SYK P43405 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CNR1 P21554 1/20 0.37
GPR35 Q9HC97 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8468606 0.82 NPC1 (0.40) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL8322376 0.78 SMN1; SMN2 (0.49) NPC1RAB9ASMN1; SMN2GAAGRM1
Water SCHEMBL8466755 0.74 NPC1 (0.42) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL8324852 0.73 GAA (0.53) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL8328108 0.72 MAPT (0.40) RAB9AADORA3ADORA2AESR2SYK
SCHEMBL10049725 0.71 NPC1 (0.49) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL8321754 0.69 KDM4E (0.41) SMN1; SMN2GAACA9LMNAADORA3
SCHEMBL12253498 0.68 GAA (0.67) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL25253396 0.68 GAA (0.57) NPC1RAB9ASMN1; SMN2GAACA9
SCHEMBL29405629 0.68 GAA (0.57) NPC1RAB9ASMN1; SMN2GAACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP disclosed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO disclosed