SCHEMBL8322376

SCHEMBL8322376

Oc1c2ncc3ccccc3c2nn1-c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
LMNA P02545 1/20 0.49
GABRA1 P14867 6/20 0.42
GABRA2 P47869 6/20 0.42
GAA P10253 2/20 0.40
ESR2 Q92731 1/20 0.38
GRM1 Q13255 2/20 0.38
GRM5 P41594 1/20 0.38
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
PLA2G10 O15496 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8462048 0.86 KDM4E (0.39) SMN1; SMN2NPC1RAB9ALMNAESR2
SCHEMBL8321754 0.86 KDM4E (0.41) SMN1; SMN2LMNAGAAADORA3ADORA2A
SCHEMBL8320446 0.86 NPC1 (0.49) SMN1; SMN2NPC1RAB9ALMNAGABRA1
SCHEMBL8466300 0.85 GAA (0.43) SMN1; SMN2NPC1RAB9ALMNAGAA
SCHEMBL8324694 0.83 MAPT (0.40) RAB9AADORA3NPSR1
SCHEMBL8322673 0.83 AURKA (0.36) SMN1; SMN2NPC1RAB9ALMNAGAA
SCHEMBL8466029 0.81 SCN9A (0.32) SMN1; SMN2NPC1RAB9ALMNANPSR1
SCHEMBL8329043 0.80 TEAD1 (0.39) SMN1; SMN2
SCHEMBL8319903 0.79 GABRA1 (0.37) SMN1; SMN2NPC1RAB9ALMNAGABRA1
SCHEMBL8326878 0.78 KDM4E (0.41) GAAADORA3ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP disclosed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO disclosed