SCHEMBL8524484

SCHEMBL8524484

Cc1ccc(-c2csc(-c3ccncc3)n2)c2c1CCCC(=O)N2C(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CDK5 Q00535 14/20 0.38
CDK5R1 Q15078 14/20 0.38
CYP19A1 P11511 2/20 0.38
AR P10275 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP17A1 P05093 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523986 0.85 CDK5 (0.40) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8525334 0.80 CDK5 (0.39) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8525624 0.76 CDK5 (0.41) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8525097 0.74 CDC25A (0.46) KDM4ENPC1RAB9ASMN1; SMN2CYP19A1
SCHEMBL8524244 0.72 CDK5 (0.38) KDM4ENPC1RAB9ASMN1; SMN2CDK5
Hydrochloric Acid SCHEMBL8524829 0.71 CYP19A1 (0.48) KDM4ENPC1RAB9ASMN1; SMN2CYP19A1
SCHEMBL8523719 0.69 CDK5 (0.44) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8484367 0.67 CDC25A (0.48) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8525207 0.67 KDM4E (0.42) KDM4ENPC1RAB9ASMN1; SMN2CDK5
SCHEMBL8483824 0.66 CDC25A (0.56) KDM4ENPC1RAB9ASMN1; SMN2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed