SCHEMBL8524730

SCHEMBL8524730

CC(NC(=O)CNc1ccc2c(C(=O)NCc3ccc(C#N)cc3)cccc2c1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
AKR1B1 P15121 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
FNTA P49354 3/20 0.39
FNTB P49356 3/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525059 0.82 HDAC2 (0.46) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8494353 0.76 HDAC2 (0.55) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL1320296 0.75 HDAC2 (0.50) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8525436 0.75 HDAC2 (0.50) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8525574 0.73 AKR1B1 (0.48) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL1110102 0.71 TUBB (0.46) CA12CA1CA2CA7AKR1B1
SCHEMBL8524189 0.71 AKR1B1 (0.48) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8524259 0.71 AKR1B1 (0.39) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL1110380 0.69 AKR1B1 (0.40) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8525044 0.69 PKLR (0.49) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed