SCHEMBL8525246

SCHEMBL8525246

C=CC([N]c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
LMNA P02545 1/20 0.34
CYP3A4 P08684 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
ALOX15 P16050 2/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TSHR P16473 2/20 0.32
DPP4 P27487 2/20 0.32
F2 P00734 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3261585 0.79 CYP2C19 (0.36) ALDH1A1LMNACYP3A4KDM4EMAPT
SCHEMBL3258485 0.76 KDM4E (0.40) ALDH1A1LMNACYP3A4KDM4EMAPT
SCHEMBL10452869 0.72 CYP2C19 (0.36) ALDH1A1LMNACYP3A4KDM4EMAPT
SCHEMBL11766335 0.72 CYP2D6 (0.37) ALDH1A1LMNACYP3A4KDM4EMAPT
SCHEMBL30104386 0.71 CYP3A4 (0.33) ALDH1A1CYP3A4KDM4EMAPTALOX15
SCHEMBL15295377 0.71 CYP3A4 (0.33) ALDH1A1CYP3A4KDM4EMAPTALOX15
SCHEMBL488830 0.71 CYP2C19 (0.39) ALDH1A1CYP3A4KDM4EMAPTALOX15
SCHEMBL1047388 0.71 CYP2C19 (0.35) ALDH1A1LMNACYP3A4KDM4EMAPT
SCHEMBL6889278 0.71 MIF (0.34) ALDH1A1CYP3A4KDM4EMAPTALOX15
SCHEMBL30104387 0.71 CYP3A4 (0.33) ALDH1A1CYP3A4KDM4EMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005112-A REACTING SUBSTITUTED OR UNSUBSTITUTED PYRIDINE METAL COMPOUND WITH SUBSTITUTED ISOCYANATE OR ISOTHIOCYANATE KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1999-12-21 US disclosed
EP-0881217-A1 PROCESS FOR PRODUCING PYRIDINECARBOXAMIDES OR THIOCARBOXAMIDES KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1998-12-02 EP disclosed
US-4195092-A INSECTICIDES FOR TREATING MEXICAN BEAN BEETLE ELI LILLY AND COMPANY (US) 1980-03-25 US disclosed