SCHEMBL8525664

SCHEMBL8525664

CC1Cc2ccc(I)cc2N1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.38
CREBBP Q92793 2/20 0.38
TSHR P16473 1/20 0.38
EP300 Q09472 1/20 0.38
PNMT P11086 7/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
ADRA2A P08913 2/20 0.37
ADRA2B P18089 2/20 0.37
ADRA2C P18825 2/20 0.37
TDP2 O95551 1/20 0.37
AR P10275 2/20 0.35
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920989 0.78 ACHE (0.43) BRD4CREBBPTSHREP300PNMT
SCHEMBL21782466 0.78 ACHE (0.43) BRD4CREBBPTSHREP300PNMT
SCHEMBL2997969 0.76 ACHE (0.44) BRD4CREBBPTSHREP300PNMT
SCHEMBL94115 0.76 ESR2 (0.49) BRD4CREBBPTSHREP300LMNA
SCHEMBL7897325 0.76 CMA1 (0.43) BRD4CREBBPTSHREP300ADRA2A
SCHEMBL7037554 0.76 MAPT (0.42) BRD4CREBBPTSHREP300PNMT
SCHEMBL12965849 0.75 AR (0.45) BRD4CREBBPTSHREP300PNMT
SCHEMBL12965982 0.73 AR (0.44) BRD4CREBBPTSHREP300PNMT
SCHEMBL13799420 0.73 ACHE (0.47)
SCHEMBL9972552 0.73 PARP1 (0.38) BRD4CREBBPTSHREP300PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083170-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-06-21 WO disclosed
EP-2455376-A1 Heterocyclic compounds as inhibitors of hepatitis C virus (HCV) Abbott Laboratories (US) 2012-05-23 EP disclosed
WO-2010144646-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-12-16 WO disclosed
WO-2010120935-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-10-21 WO disclosed