Benzenesulfonamide

Benzenesulfonamide

SCHEMBL8525970

NS(=O)(=O)c1ccccc1.O=S(=O)(Nc1cccn1-c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.50

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 2/20 0.50
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
KIF11 P52732 1/20 0.44
PTGS2 P35354 6/20 0.44
PTGS1 P23219 4/20 0.44
OXTR P30559 2/20 0.43
AVPR1A P37288 2/20 0.43
HSD11B1 P28845 1/20 0.42
ACLY P53396 1/20 0.41
MAPT P10636 1/20 0.41
AVPR2 P30518 1/20 0.41
GPR27 Q9NS67 1/20 0.41
EPHX2 P34913 2/20 0.41
PPARG P37231 1/20 0.41
NR1H3 Q13133 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8505556 0.94 OXTR (0.48) PTGES2OXTRAVPR1AHSD11B1ACLY
Benzenesulfonamide SCHEMBL8524570 0.85 CA12 (0.48) PTGES2CA12CA1CA2CA9
Benzenesulfonamide SCHEMBL8525288 0.85 CA12 (0.48) CA12CA1CA2CA9PTGS2
Benzenesulfonamide SCHEMBL8525761 0.85 CA1 (0.48) CA12CA1CA2CA9PTGS2
SCHEMBL8503384 0.81 CYP2C9 (0.54) CYP2C9ALDH1A1LMNA
Benzenesulfonamide SCHEMBL8526038 0.81 PTGES2 (0.48) PTGES2CA12CA1CA2CA9
Benzenesulfonamide SCHEMBL8525643 0.80 CA1 (0.46) CA12CA1CA2CA9PTGS2
SCHEMBL8506074 0.78 CYP2C9 (0.52) MAPTCYP2C9ALDH1A1LMNA
SCHEMBL8504924 0.78 CYP2C9 (0.52) CA12CA1CA2CA9MAPT
SCHEMBL8505905 0.78 CYP2C9 (0.51) CYP2C9ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP disclosed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO disclosed