Benzenesulfonamide

Benzenesulfonamide

SCHEMBL8526038

Cc1ccc(NS(=O)(=O)c2ccccc2)n1-c1ccc(C(F)(F)F)cc1.NS(=O)(=O)c1ccccc1

nearest known ligand 0.48

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Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 2/20 0.48
PTGS2 P35354 6/20 0.46
OXTR P30559 3/20 0.44
AVPR1A P37288 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
KIF11 P52732 1/20 0.43
PTGS1 P23219 4/20 0.42
HSD11B1 P28845 2/20 0.42
FFAR4 Q5NUL3 1/20 0.40
EPHX2 P34913 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8506143 0.94 PTGS2 (0.50) PTGES2PTGS2OXTRAVPR1AHSD11B1
Benzenesulfonamide SCHEMBL8526332 0.84 CA12 (0.47) CA1CA2CA12CA9
Benzenesulfonamide SCHEMBL8526469 0.82 CA1 (0.47) PTGES2PTGS2CA1CA2CA12
Benzenesulfonamide SCHEMBL8526101 0.82 POLB (0.51) PTGS2CA1CA2CA12CA9
Benzenesulfonamide SCHEMBL8525970 0.81 PTGES2 (0.50) PTGES2PTGS2OXTRAVPR1ACA1
SCHEMBL8502466 0.81 CYP2C9 (0.53) PTGS2CA1CA2CA12CA9
SCHEMBL8504469 0.80 TSHR (0.48) PTGS2OXTRFFAR4
SCHEMBL8504989 0.80 CYP2C9 (0.53) PTGS2CA1CA2CA12CA9
Benzenesulfonamide SCHEMBL8525170 0.79 PTGS1 (0.44) PTGS2CA1CA2CA12CA9
SCHEMBL8502313 0.77 ALDH1A1 (0.49) OXTRAVPR1AFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP disclosed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO disclosed