SCHEMBL8526255

SCHEMBL8526255

NC(=O)C(N)c1cc[c]cc1

nearest known ligand 0.31

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
EPHX1 P07099 1/20 0.31
GRM8 O00222 1/20 0.31
GRM6 O15303 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
DRD3 P35462 1/20 0.31
GRM4 Q14833 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27397292 0.82 HSD17B10 (0.47) MEN1CYP2D6CYP2C9CYP2C19KMT2A
SCHEMBL3535148 0.82 BRD4 (0.32) MEN1CYP2D6CYP2C9CYP2C19KMT2A
Hydrochloric Acid SCHEMBL27583753 0.77 EPHX1 (0.47) CYP2D6EPHX1DPP4
SCHEMBL17140609 0.77 LMNA (0.38) EPHX1
SCHEMBL16935655 0.77
SCHEMBL5144744 0.77
SCHEMBL544671 0.76 EPHX1 (0.50) CYP2D6EPHX1DPP4
SCHEMBL2332933 0.76 EPHX1 (0.50) CYP2D6EPHX1DPP4
SCHEMBL1218849 0.76 EPHX1 (0.50) CYP2D6EPHX1DPP4
SCHEMBL10822383 0.76 EPHX1 (0.53) CYP2C9EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1326440-A Piperdine CCR-3 receptor antagonists HOFFMANN LA ROCHE (CH) 2001-12-12 CN claimed
CN-1326440-A Piperdine CCR-3 receptor antagonists HOFFMANN LA ROCHE (CH) 2001-12-12 CN disclosed
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed