SCHEMBL8526299

SCHEMBL8526299

CCOC(CNc1ccc(C)c(Cl)c1)OCC

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.47
HPGD P15428 3/20 0.47
MAPT P10636 9/20 0.45
SMN1; SMN2 Q16637 5/20 0.43
AGTR1 P30556 3/20 0.43
GAA P10253 2/20 0.43
NPC1 O15118 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
RAB9A P51151 2/20 0.42
CYP2C9 P11712 1/20 0.42
RAPGEF4 Q8WZA2 1/20 0.41
LMNA P02545 2/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
EPHX1 P07099 1/20 0.40
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3084018 0.81 ALDH1A1 (0.38) ALDH1A1MAPTSMN1; SMN2GAANPC1
SCHEMBL11070949 0.78 EPHX1 (0.44) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL5713058 0.76 MAPT (0.48) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL13359814 0.76 ALDH1A1 (0.49) ALDH1A1HPGDMAPTSMN1; SMN2AGTR1
SCHEMBL1798419 0.76 ALDH1A1 (0.53) ALDH1A1HPGDMAPTSMN1; SMN2AGTR1
SCHEMBL24307977 0.74 MAPT (0.55) ALDH1A1HPGDMAPTGAACYP1A2
SCHEMBL13326762 0.74 ALDH1A1 (0.49) ALDH1A1HPGDMAPTSMN1; SMN2AGTR1
SCHEMBL131784 0.73 EPHX1 (0.61) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL5608579 0.71 HTT (0.51) ALDH1A1MAPTSMN1; SMN2GAACYP1A2
SCHEMBL935506 0.71 MAPT (0.49) ALDH1A1MAPTSMN1; SMN2GAAEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834494-A SEROTONIN 5HT2B/2C RECEPTOR ANTAGONISTS; CNS NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS; IRRITABLE BOWEL SYNDROME SMITHKLINE BEECHAM P.L.C. (GB) 1998-11-10 US disclosed
EP-0707581-B1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-02-26 EP disclosed
EP-0707581-A1 INDOLINE DERIVATIVES AS 5HT 2C? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-24 EP disclosed
WO-1995001976-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-01-19 WO disclosed