SCHEMBL8526529

SCHEMBL8526529

COc1ccc2c(c1OC)CC[C@]2(N)C(C)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
PDE4A P27815 2/20 0.40
NQO2 P16083 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ABCB1 P08183 3/20 0.35
ACHE P22303 1/20 0.35
LMNA P02545 2/20 0.34
CYP3A4 P08684 1/20 0.34
HSP90AA1 P07900 2/20 0.34
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL355655 0.81 PARP1 (0.40) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL10723706 0.77 ALDH1A1 (0.46) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL27371146 0.73 KDM4E (0.50) PARP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL11006912 0.72 PARP1 (0.43) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL7655996 0.70 KDM4E (0.40) ALDH1A1KDM4EHPGDPDE4AMTNR1A
SCHEMBL12379988 0.70 ABCB1 (0.45) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL28054318 0.69 ADRA1A (0.38) ALDH1A1KDM4EHPGDMTNR1AMTNR1B
SCHEMBL11083684 0.68 PARP1 (0.41) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL11027320 0.65 PARP1 (0.41) PARP1ALDH1A1KDM4EHPGDPDE4A
SCHEMBL2468652 0.64 KDM4E (0.44) ALDH1A1KDM4EMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877218-A PARKINSON'S DISEASE; ANTIEPILEPSY AGENTS; ANTICONVULSANTS TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 1999-03-02 US claimed
WO-1999033858-A9 ESTRONE SULFAMATE INHIBITORS OF ESTRONE SULFATASE, AND ASSOCIATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE STANFORD RES INST INT (US) 1999-10-28 WO disclosed