SCHEMBL8526563

SCHEMBL8526563

CCOc1c(C)ccc(C(=O)S)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 2/20 0.35
SCN5A Q14524 1/20 0.35
HCRTR1 O43613 1/20 0.35
PLK1 P53350 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303456 0.79 ADORA3 (0.35) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL8526566 0.77 SCN5A (0.36) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL9303460 0.76 SCN5A (0.35) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL6985548 0.75 NQO1 (0.42) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL8680142 0.75 HTT (0.33) ALDH1A1TSHRMEN1KMT2ASMN1; SMN2
SCHEMBL28452343 0.73 ALDH1A1 (0.36) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL28274071 0.73 HSD17B10 (0.48) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL28127002 0.72 ALDH1A1 (0.40) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL10434028 0.72 NQO1 (0.48) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL28126645 0.71 TSHR (0.55) ALDH1A1HSD17B10L3MBTL1TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639173-B1 CERTAIN 2-(2'METHYL-3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA LTD (GB) 1998-03-11 EP disclosed
EP-0639173-A1 CERTAIN 2-(2'METHYL-3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA LIMITED (GB) 1995-02-22 EP disclosed
US-5329041-A For herbicides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-07-12 US disclosed
EP-0639173-A4 CERTAIN 2-(2'METHYL-3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES. ZENECA LTD (GB) 1993-09-17 EP disclosed
WO-1992012957-A1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES NGUYEN NHAN H (US) 1992-08-06 WO disclosed
WO-1992012953-A1 CERTAIN 2-(2'METHYL-3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA LIMITED (GB) 1992-08-06 WO disclosed
US-5110979-A Trisubstituted benzoic acid intermediates IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-05 US disclosed