SCHEMBL8527587

SCHEMBL8527587

O=C(Nc1ccc(Br)c(C(F)(F)F)c1)C(F)(F)F

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.64
LMNA P02545 4/20 0.64
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
NPSR1 Q6W5P4 2/20 0.64
XBP1 P17861 1/20 0.64
HTT P42858 3/20 0.61
EPHX1 P07099 2/20 0.61
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
SMN1; SMN2 Q16637 2/20 0.59
TMPRSS4 Q9NRS4 1/20 0.56
TAS2R14 Q9NYV8 1/20 0.52
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
KDR P35968 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8407479 0.86 AR (0.63) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL8409105 0.84 MAPT (0.59) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL8903304 0.84 CYP1A2 (0.54) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL8902443 0.84 CYP1A2 (0.54) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL30977691 0.83 EPHX1 (0.74) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL1431941 0.83 EPHX1 (0.74) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL2705806 0.83 MAPT (0.64) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL8410666 0.82 EPHX1 (0.60) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL8530877 0.81 AR (0.58) SMN1; SMN2CYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL29535627 0.81 CYP1A2 (0.51) MAPTLMNAMEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596358-B1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1998-10-28 EP disclosed
US-5484953-A CHEMICAL INTERMEDIATES FOR BENZIMIDAZOLES FOR INSECTICIDES OR NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-01-16 US disclosed
EP-0596358-A1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1994-05-11 EP disclosed