SCHEMBL8528103

SCHEMBL8528103

COCc1cc(C(=O)O)ccc1-c1ccc(N2CCCC2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
IP6K1 Q92551 1/20 0.50
IP6K3 Q96PC2 1/20 0.50
IP6K2 Q9UHH9 1/20 0.50
HPGD P15428 7/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
TSHR P16473 3/20 0.47
LMNA P02545 1/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
RXFP1 Q9HBX9 1/20 0.47
PRKAB2 O43741 1/20 0.46
PRKAG1 P54619 1/20 0.46
PRKAA2 P54646 1/20 0.46
PRKAA1 Q13131 1/20 0.46
PRKAG3 Q9UGI9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8140892 0.84 PKM (0.52) ALDH1A1HPGDTSHRLMNANPC1
SCHEMBL792262 0.82 MAPT (0.42) ALDH1A1HPGDLMNANPC1RAB9A
SCHEMBL13286265 0.82 CHEK1 (0.42) ALDH1A1HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL792229 0.80 CHEK1 (0.41) ALDH1A1HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL13286254 0.79 CHEK1 (0.39) HPGDTSHRLMNA
SCHEMBL792246 0.79 F10 (0.44) ALDH1A1LMNANPC1RAB9APRKAB2
SCHEMBL22575179 0.77 SMN1; SMN2 (0.41) ALDH1A1HPGDTSHRLMNANPC1
SCHEMBL6715880 0.77 RARB (0.45) ALDH1A1TSHRLMNANPC1RAB9A
SCHEMBL27736080 0.76 EGFR (0.53) ALDH1A1
SCHEMBL8135917 0.76 ALDH1A1 (0.58) ALDH1A1IP6K1IP6K3IP6K2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888358-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1999-01-07 EP disclosed
WO-1997034901-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 1997-09-25 WO disclosed