SCHEMBL8528518

SCHEMBL8528518

COC(=O)CN(CC(=O)OC)C(=O)Cc1ccc(CN(C(=O)C(c2ccccc2)c2ccccc2)[C@H](CCCNC(=N)N)C(N)=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
EPOR P19235 4/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
CNR1 P21554 1/20 0.32
ALOX5 P09917 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
PRSS1 P07477 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528680 0.91 TDP1 (0.36) TDP1EPORHDAC1HDAC7CNR1
SCHEMBL8529309 0.86 CNR1 (0.36) TDP1CNR1MEN1KMT2AF2
SCHEMBL7039838 0.86 TDP1 (0.36) TDP1CNR1MEN1KMT2AITGB3
SCHEMBL7750689 0.86 MEN1 (0.42) TDP1CNR1MEN1KMT2AF2
SCHEMBL7039868 0.86 ITGB3 (0.33) TDP1EPORHDAC1HDAC7CNR1
SCHEMBL6901612 0.85 CNR1 (0.43) TDP1HDAC1HDAC7CNR1KMT2A
SCHEMBL30905434 0.85 CNR1 (0.41) TDP1EPORCNR1MEN1KMT2A
SCHEMBL1389118 0.85 CNR1 (0.41) TDP1EPORCNR1MEN1KMT2A
SCHEMBL8121296 0.84 F2 (0.38) TDP1MEN1KMT2AF2F10
SCHEMBL4651831 0.84 CNR1 (0.42) TDP1EPORCNR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed