SCHEMBL8529428

SCHEMBL8529428

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](COC(=O)C(C)C)[C@@H](O)[C@@H]1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HINT1 P49773 3/20 0.61
NT5E P21589 2/20 0.53
ADORA3 P0DMS8 3/20 0.52
CYP2C19 P33261 1/20 0.52
SLC29A1 Q99808 3/20 0.52
ADORA2A P29274 3/20 0.51
ADORA2B P29275 3/20 0.51
ADORA1 P30542 1/20 0.51
MARS1 P56192 1/20 0.51
CCNT1 O60563 1/20 0.49
CCNK O75909 1/20 0.49
CDK7 P50613 1/20 0.49
CDK9 P50750 1/20 0.49
CCNH P51946 1/20 0.49
MNAT1 P51948 1/20 0.49
CDK12 Q9NYV4 1/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA4 P22748 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530562 0.90 HINT1 (0.62) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL8529529 0.89 HINT1 (0.63) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL15643631 0.87 ADORA3 (0.67) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL16141624 0.87 ADORA3 (0.67) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL8532674 0.87 HINT1 (0.61) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL8532886 0.87 HINT1 (0.61) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL25354772 0.86 HINT1 (0.62) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL8529229 0.85 HINT1 (0.59) HINT1NT5EADORA3CYP2C19SLC29A1
SCHEMBL8760103 0.84 HINT1 (0.58) HINT1NT5EADORA3CYP2C19SLC29A1
Nelarabine SCHEMBL13575801 0.84 CYP2C19 (0.71) NT5EADORA3CYP2C19SLC29A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US claimed
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed