SCHEMBL8529435

SCHEMBL8529435

S=C1CSc2cccc(Cl)c2CN1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
PNMT P11086 1/20 0.38
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
PSMB8 P28062 2/20 0.31
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
HSD17B3 P37058 1/20 0.31
PIM1 P11309 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8527294 0.80 ALDH1A1 (0.42) ALDH1A1HDAC8
SCHEMBL8526839 0.80 HPGD (0.39) ALDH1A1PNMTHSD17B3PIM1
SCHEMBL7555387 0.76 PNMT (0.32) PNMTHSD17B3
SCHEMBL7555383 0.76 PNMT (0.32) PNMTHSD17B3
SCHEMBL7554811 0.73 MAPK14 (0.31)
SCHEMBL7562688 0.73 ATM (0.43) ALDH1A1MEN1KMT2AHSD17B3
SCHEMBL7554807 0.73 MAPK14 (0.31)
SCHEMBL11272845 0.72 ALDH1A1 (0.53) ALDH1A1PSMB8HSD17B3PIM1HDAC4
SCHEMBL8530034 0.72 ALDH1A1 (0.52) ALDH1A1MEN1POLBKMT2AHSD17B3
SCHEMBL7554455 0.69 RYR2 (0.53) ALDH1A1PNMTMEN1KMT2AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0667866-B1 1,4-BENZOTHIAZEPINES USEFUL AS NEUROLOGICAL AGENTS KNOLL AG (DE) 1998-03-11 EP disclosed
US-5580866-A Therapeutic 1,4-thiazepines THE BOOTS COMPANY PLC (GB) 1996-12-03 US disclosed
EP-0667866-A1 1,4-BENZOTHIAZEPINES USEFUL AS NEUROLOGICAL AGENTS Knoll AG (DE) 1995-08-23 EP disclosed
WO-1994011360-A1 1,4-BENZOTHIAZEPINES USEFUL AS NEUROLOGICAL AGENTS THE BOOTS COMPANY PLC (GB) 1994-05-26 WO disclosed