SCHEMBL8529693

SCHEMBL8529693

CC1CCC(c2ccc(C(=O)N=C(N)N)c(C(F)(F)C(F)(F)F)c2S(C)(=O)=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 12/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
ADRA1D P25100 1/20 0.37
HTR2A P28223 1/20 0.37
SLC6A3 Q01959 1/20 0.37
SLC9A2 Q9UBY0 1/20 0.37
KCNH2 Q12809 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533030 0.84 SLC9A1 (0.42) SLC9A1CYP3A4
SCHEMBL8533178 0.83 SLC9A1 (0.45) SLC9A1
SCHEMBL8585538 0.82 ALDH1A1 (0.36)
SCHEMBL8533216 0.81 SLC9A1 (0.47) SLC9A1CYP3A4
SCHEMBL8528602 0.80 SLC9A1 (0.41) SLC9A1
SCHEMBL8529433 0.80 SLC9A1 (0.48) SLC9A1CYP3A4CYP2C9CYP2C19
SCHEMBL8580832 0.79 SLC9A1 (0.45) SLC9A1CYP3A4
SCHEMBL8528555 0.78 SLC9A1 (0.48) SLC9A1
SCHEMBL8530489 0.78 SLC9A1 (0.46) SLC9A1CYP3A4CYP2C9CYP2C19
SCHEMBL8529686 0.77 SLC9A1 (0.52) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840761-A Alkylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-11-24 US disclosed
EP-0699663-B1 Alkyl-benzoylguanidine derivatives MERCK PATENT GMBH (DE) 1998-11-04 EP disclosed
EP-0699663-A1 Alkyl-benzoylguanidine derivatives MERCK PATENT GmbH (DE) 1996-03-06 EP disclosed