SCHEMBL8530891

SCHEMBL8530891

CCCC(=O)OC(=O)NC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.64
EPHX1 P07099 1/20 0.42
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HDAC3 O15379 4/20 0.37
HDAC1 Q13547 4/20 0.37
HDAC2 Q92769 4/20 0.37
HDAC8 Q9BY41 4/20 0.37
HDAC6 Q9UBN7 1/20 0.37
FFAR3 O14843 3/20 0.36
TSHR P16473 3/20 0.36
CTSD P07339 1/20 0.36
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CYP2D6 P10635 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRNB2 P17787 1/20 0.34
NFKB1 P19838 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27943916 0.86 EPHX1 (0.48) ALDH1A1EPHX1CES2CES1TSHR
SCHEMBL29111620 0.83 EPHX1 (0.55) ALDH1A1EPHX1CES2CES1TSHR
SCHEMBL29111622 0.83 EPHX1 (0.55) ALDH1A1EPHX1CES2CES1TSHR
SCHEMBL29111625 0.83 EPHX1 (0.55) ALDH1A1EPHX1CES2CES1TSHR
SCHEMBL27630422 0.83 EPHX1 (0.55) ALDH1A1EPHX1CES2CES1TSHR
SCHEMBL15810277 0.82
SCHEMBL28937192 0.81 ALDH1A1 (0.64) ALDH1A1CES2CES1HDAC3HDAC1
SCHEMBL13316206 0.79 CHRNB2 (0.39) ALDH1A1EPHX1TSHRCHRM2CHRM4
SCHEMBL8529427 0.79 ALDH1A1 (0.61) ALDH1A1EPHX1CES2CES1HDAC3
SCHEMBL30568759 0.79 ALDH1A1 (1.00) ALDH1A1CES2CES1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108342422-B Preparation method of N-substituted amino carbonyl ester compound and application of immobilized lipase 北京海美桐医药科技有限公司 2020-08-14 CN disclosed
CN-108342422-A The preparation method of N- substituted amido carbonyl ester type compounds and the application of immobilized lipase 北京海美桐医药科技有限公司 2018-07-31 CN disclosed
CN-104662004-B Novel rebamipide prodrug, method for producing same, and usage thereof 三进制药株式会社 2017-04-19 CN disclosed
EP-0873123-A4 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIV PITTSBURGH (US) 1999-02-03 EP disclosed
EP-0873123-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 1998-10-28 EP disclosed
WO-1997017070-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 1997-05-15 WO disclosed