SCHEMBL8530895

SCHEMBL8530895

[CH2]c1cn(C(=O)OCc2ccccc2)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.49
MAOA P21397 1/20 0.49
RCOR1 Q9UKL0 1/20 0.49
TACR3 P29371 1/20 0.46
P2RX4 Q99571 2/20 0.44
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
P2RX1 P51575 1/20 0.43
P2RX3 P56373 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
MAPK1 P28482 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530899 0.84 KDM1A (0.48) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL16399234 0.84 TACR3 (0.53) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL6283431 0.83 L3MBTL1 (0.53) ALDH1A1KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9027466 0.83 ALDH1A1 (0.49) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL2253248 0.82 TACR3 (0.51) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL9572545 0.82 KDM1A (0.57) KDM1AMAOARCOR1TACR3ALDH1A1
SCHEMBL31186285 0.81 STAT3 (0.52) KDM1AMAOARCOR1TACR3ALDH1A1
SCHEMBL9116988 0.80 TACR3 (0.49) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL2253255 0.80 ALDH1A1 (0.49) KDM1AMAOARCOR1TACR3P2RX4
SCHEMBL10845805 0.80 KDM1A (0.45) KDM1AMAOARCOR1TACR3P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0460679-B1 Endothelin antagonistic peptide derivatives BANYU PHARMA CO LTD (JP) 1998-10-28 EP disclosed
US-5691315-A CARDIOVASCULAR DISORDERS; VASODILATOR; BRONCHODILATOR BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5470833-A Vasodilators, bronchodilators BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-11-28 US disclosed
US-5444152-A Vasolidator or bronchodilator BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-22 US disclosed
EP-0460679-A2 Endothelin antagonistic peptide derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-12-11 EP disclosed