SCHEMBL8530934

SCHEMBL8530934

Cc1cn(CC(=O)OC(C)(C)C)c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
ALDH1A1 P00352 8/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 3/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
KDM4E B2RXH2 2/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TSHR P16473 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530927 0.84 GAA (0.49) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL8531844 0.84 GAA (0.69) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL17023509 0.83 GAA (0.58) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL8528645 0.82 ALDH1A1 (0.71) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL8598898 0.82 ALDH1A1 (0.70) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL19208816 0.82 GAA (0.56) KMT2AALDH1A1GAALMNAPOLB
SCHEMBL10165370 0.82 KMT2A (0.66) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL12479405 0.82 LMNA (0.68) KMT2AALDH1A1GAAMAPTLMNA
SCHEMBL19208559 0.80 KDM4E (0.68) KMT2AALDH1A1GAALMNAPOLB
SCHEMBL5956307 0.80 GAA (0.54) MEN1KMT2AALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0460679-B1 Endothelin antagonistic peptide derivatives BANYU PHARMA CO LTD (JP) 1998-10-28 EP disclosed
US-5691315-A CARDIOVASCULAR DISORDERS; VASODILATOR; BRONCHODILATOR BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5470833-A Vasodilators, bronchodilators BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-11-28 US disclosed
US-5444152-A Vasolidator or bronchodilator BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-22 US disclosed
EP-0460679-A2 Endothelin antagonistic peptide derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-12-11 EP disclosed