SCHEMBL8533002

SCHEMBL8533002

CCOc1ccc2nc(NC(=O)CN3CCN(c4ccc(C(C)=O)cc4)CC3)sc2c1

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.70
LMNA P02545 2/20 0.70
USP2 O75604 1/20 0.70
TSHR P16473 1/20 0.70
LRRK2 Q5S007 2/20 0.67
ALDH1A1 P00352 3/20 0.60
KDM4E B2RXH2 1/20 0.60
POLB P06746 2/20 0.59
KMT2A Q03164 2/20 0.59
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
HSD17B10 Q99714 1/20 0.58
TP53 P04637 2/20 0.57
HTT P42858 2/20 0.57
MAPK1 P28482 1/20 0.57
MEN1 O00255 1/20 0.56
MAPT P10636 1/20 0.56
CLK1 P49759 1/20 0.55
SLC27A1 Q6PCB7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11266059 0.85 SLC27A1 (0.60) SMN1; SMN2ALDH1A1POLBKMT2AHTT
SCHEMBL8354249 0.84 SMN1; SMN2 (0.71) SMN1; SMN2LMNAUSP2TSHRLRRK2
SCHEMBL8354375 0.82 SMN1; SMN2 (0.68) SMN1; SMN2LMNAUSP2TSHRLRRK2
Hydrochloric Acid SCHEMBL8353865 0.82 SMN1; SMN2 (0.67) SMN1; SMN2LMNAUSP2TSHRLRRK2
SCHEMBL8354234 0.81 ALDH1A1 (0.76) SMN1; SMN2LMNAUSP2TSHRALDH1A1
SCHEMBL21753691 0.80 LRRK2 (1.00) SMN1; SMN2LMNAUSP2LRRK2ALDH1A1
SCHEMBL30620435 0.79 SMN1; SMN2 (0.63) SMN1; SMN2LMNAUSP2TSHRALDH1A1
SCHEMBL27008579 0.79 SMN1; SMN2 (0.63) SMN1; SMN2LMNAUSP2TSHRALDH1A1
SCHEMBL8350371 0.79 SLC27A1 (0.68) LMNAALDH1A1KDM4EPOLBKMT2A
SCHEMBL8356375 0.79 ALDH1A1 (0.75) SMN1; SMN2LMNAUSP2TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031096-A1 PIPERAZINE DERIVATIVES USEFUL AS HYPOGLYCEMIC AGENTS SHAMAN PHARMACEUTICALS, INC. (US) 1999-06-24 WO disclosed