SCHEMBL8533857

SCHEMBL8533857

CC(C)CNc1ccc2c(ccn2-c2ccc(OCC3CCN(C(=O)OC(C)C)CC3)cn2)c1

nearest known ligand 0.55

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533856 0.89 GPR119 (0.55) GPR119
SCHEMBL9253174 0.81 GPR119 (0.53) GPR119
SCHEMBL9248533 0.80 GPR119 (0.45) GPR119
SCHEMBL8537262 0.75 GPR119 (0.53) GPR119
SCHEMBL9263416 0.74 GPR119 (0.59) GPR119
SCHEMBL9266545 0.74 GPR119 (0.50) GPR119
SCHEMBL11956857 0.74 GPR119 (0.84) GPR119
SCHEMBL8533540 0.74 GPR119 (0.45) GPR119
SCHEMBL15253175 0.74 GPR119 (0.53) GPR119
SCHEMBL9260951 0.72 GPR119 (0.56) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2643311-A1 BICYCLIC GPR119 MODULATORS Lupin Limited (IN) 2013-10-02 EP disclosed
WO-2012069917-A1 BICYCLIC GPR119 MODULATORS LUPIN LIMITED (IN) 2012-05-31 WO disclosed