SCHEMBL8534112

SCHEMBL8534112

Nc1cc2cccc(O)c2cc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.61
CTDSP1 Q9GZU7 1/20 0.61
CYP1A2 P05177 1/20 0.50
GRIN2D O15399 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRIN2B Q13224 1/20 0.50
GRIN2C Q14957 1/20 0.50
HSD17B1 P14061 5/20 0.47
HSD17B2 P37059 5/20 0.47
ESR1 P03372 2/20 0.47
ESR2 Q92731 2/20 0.47
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
IDO1 P14902 2/20 0.42
TDO2 P48775 1/20 0.42
HDAC3 O15379 1/20 0.41
EP300 Q09472 1/20 0.41
KAT2B Q92831 1/20 0.41
KAT8 Q9H7Z6 1/20 0.41
NCOR2 Q9Y618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10713270 0.84 PLAU (0.59) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL2115683 0.83 CYP1A2 (0.62) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL29857010 0.83 CYP1A2 (0.62) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL430311 0.80 CYP1A2 (0.59) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL30323818 0.80 CYP1A2 (0.59) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL9331048 0.79 AURKA (0.53) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL10796264 0.79 GRIN2D (0.67) PLAUCTDSP1GRIN2DGRIN2AGRIN2B
SCHEMBL3316203 0.78 CYP1A2 (0.56) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL30994717 0.78 CYP1A2 (0.56) PLAUCTDSP1CYP1A2GRIN2DGRIN2A
SCHEMBL7754286 0.78 ALDH1A1 (0.56) PLAUCYP1A2ALOX15TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776931-A TREATING PHYSIOLOGICAL DISORDER ASSOCIATED WITH EXCESS OF NEUROPEPTIDE Y ELI LILLY AND COMPANY (US) 1998-07-07 US disclosed
US-5093495-A Benzoheterocyclic compounds SHELL OIL COMPANY (US) 1992-03-03 US disclosed
US-5071996-A Benzheterocyclic compounds SHELL OIL COMPANY (US) 1991-12-10 US disclosed