SCHEMBL853489

SCHEMBL853489

CCOC(=O)C1CCN(CCN)CC1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.55
LMNA P02545 2/20 0.53
KCNH2 Q12809 3/20 0.53
ALDH1A1 P00352 6/20 0.53
TDP1 Q9NUW8 1/20 0.51
KDM4E B2RXH2 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
LTA4H P09960 1/20 0.50
POLB P06746 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8479751 0.98 MAPT (0.54) MAPTLMNAKCNH2ALDH1A1TDP1
SCHEMBL15569388 0.90 MAPT (0.62) MAPTLMNAKCNH2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6751953 0.89 KCNH2 (0.55) MAPTLMNAKCNH2ALDH1A1TDP1
SCHEMBL4172495 0.86 MAPT (0.58) MAPTLMNAKCNH2ALDH1A1KDM4E
SCHEMBL15956633 0.85 MAPT (0.57) MAPTLMNAKCNH2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL5071255 0.85 MAPT (0.57) MAPTLMNAKCNH2ALDH1A1KDM4E
SCHEMBL17284705 0.84 MAPT (0.53) MAPTLMNAKCNH2ALDH1A1KDM4E
SCHEMBL1440000 0.83 MAPT (0.55) MAPTLMNAKCNH2ALDH1A1KDM4E
SCHEMBL30924929 0.83 MAPT (0.55) MAPTLMNAKCNH2ALDH1A1KDM4E
SCHEMBL30414662 0.83 MAPT (0.55) MAPTLMNAKCNH2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119968375-A Heterocyclic derivatives as Janus kinase inhibitors 奇斯药制品公司 2025-05-09 CN disclosed
WO-2023122298-A1 PROTEIN STABILIZING COMPOUNDS CONTAINING USP28 AND/OR USP25 TARGETING LIGANDS Stablix, Inc. (US) 2023-06-29 WO disclosed
EP-3564240-A1 PIPERIDINE INTERMEDIATES Purdue Pharma L.P. (US) 2019-11-06 EP disclosed
US-9527840-B2 Substituted-quinoxaline-type piperidine compounds and the uses thereof PURDUE PHARMA L.P. (US) 2016-12-27 US disclosed
US-9527840-B2 Substituted-quinoxaline-type piperidine compounds and the uses thereof PURDUE PHARMA L.P. (US) 2016-12-27 US disclosed
US-9527840-B2 Substituted-quinoxaline-type piperidine compounds and the uses thereof PURDUE PHARMA L.P. (US) 2016-12-27 US disclosed
EP-3101018-A1 SUBSTITUTED-QUINOXALINE-TYPE-PIPERIDINE COMPOUNDS AND THE USES THEREOF Purdue Pharma L.P. (US) 2016-12-07 EP disclosed
EP-3101018-A1 SUBSTITUTED-QUINOXALINE-TYPE-PIPERIDINE COMPOUNDS AND THE USES THEREOF Purdue Pharma L.P. (US) 2016-12-07 EP disclosed
EP-2433937-B1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof PURDUE PHARMA LP (US) 2016-06-29 EP disclosed
EP-2433937-B1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof PURDUE PHARMA LP (US) 2016-06-29 EP disclosed
EP-2433937-A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof Purdue Pharma LP (US) 2012-03-28 EP disclosed
WO-2011008247-A1 FLAVIN DERIVATIVES BIORELIX, INC. (US) 2011-01-20 WO disclosed
US-20100216726-A1 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof PURDUE PHARMA L.P. (US) 2010-08-26 US disclosed
US-20100216726-A1 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof PURDUE PHARMA L.P. (US) 2010-08-26 US disclosed
US-20100216726-A1 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof PURDUE PHARMA L.P. (US) 2010-08-26 US disclosed
WO-2009027820-A2 SUBSTITUTED-QUINOXALINE-TYPE-PIPERIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA L.P. (DE) 2009-03-05 WO disclosed
US-5922717-A ANTICOAGULANTS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
CN-1024667-C process for preparing substituted aminomethyl tetralins and substituted aminomethyl hydrogenated benzopyrans and their salts BAYER AG (DE) 1994-05-25 CN disclosed
CN-1039809-A The aminomethyl tetraline that replaces and the preparation of heterocycle homologue thereof BAYER AG (DE) 1990-02-21 CN disclosed
CN-1036566-A 1,3,4,5-tetrahydro benzo [c, d] diindyl compounds BAYER AG (DE) 1989-10-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100216726-A1 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof P2RX4, P2RX5, P2RX3 MAPT 2731/4885LMNA 2734/4885KCNH2 41/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.