SCHEMBL8534932

SCHEMBL8534932

CC(C)(C)SCC(Cc1ccncc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
ERAP2 Q6P179 2/20 0.41
ERAP1 Q9NZ08 2/20 0.41
ANPEP P15144 1/20 0.41
CYP3A4 P08684 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MME P08473 1/20 0.40
KIF11 P52732 1/20 0.40
CPA1 P15085 3/20 0.39
CPA3 P15088 3/20 0.39
FOLH1 Q04609 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CPB1 P15086 1/20 0.39
CPB2 Q96IY4 1/20 0.39
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7290672 0.86 CYP1A2 (0.61) CYP1A2MMECPA1CPA3FOLH1
SCHEMBL7272157 0.86 CYP1A2 (0.61) CYP1A2MMECPA1CPA3FOLH1
SCHEMBL7438505 0.80 CYP1A2 (0.45) CYP1A2ERAP2ERAP1ANPEPCYP3A4
SCHEMBL9556401 0.79 LDHA (0.58) KIF11
SCHEMBL9556399 0.79 LDHA (0.58) KIF11
SCHEMBL7346172 0.75 CYP1A2 (0.77) CYP1A2ERAP2ERAP1ANPEPCYP3A4
SCHEMBL21896403 0.75 FOLH1 (0.51) CYP1A2ERAP2ERAP1ANPEPCPA3
SCHEMBL8531043 0.75 CYP1A2 (0.42) CYP1A2ERAP2ERAP1ANPEPCYP3A4
SCHEMBL397348 0.74 CYP1A2 (0.42) CYP1A2MMEFOLH1
SCHEMBL397349 0.74 CYP1A2 (0.42) CYP1A2MMEFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712417-A Inhibitors of retroviral proteases ABBOTT LABORATORIES (US) 1998-01-27 US disclosed
EP-0428849-A2 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-29 EP disclosed