SCHEMBL8536874

SCHEMBL8536874

CCSc1ccccc1-c1ncc[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.45
TYRO3 Q06418 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
NISCH Q9Y2I1 2/20 0.44
MTOR P42345 1/20 0.44
ADK P55263 1/20 0.44
BCHE P06276 1/20 0.44
ALOX5AP P20292 1/20 0.43
FEN1 P39748 1/20 0.43
PDE5A O76074 1/20 0.43
ALDH1A1 P00352 3/20 0.42
NPC1 O15118 2/20 0.42
KDM4E B2RXH2 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ATM Q13315 1/20 0.42
ADRA1A P35348 2/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615177 0.83 PDE5A (0.46) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8537576 0.81 CSNK1A1 (0.49) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8539114 0.81 MTOR (0.46) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL4783992 0.81 NPC1 (0.38) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8679994 0.80 CSNK1A1 (0.42) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8539546 0.80 MTOR (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8535734 0.80 TXN (0.44) CSNK1A1TYRO3DYRK1BNISCHMTOR
Hydrochloric Acid SCHEMBL20204146 0.80 CSNK1A1 (0.47) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL10583540 0.79 CYP1A2 (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8538268 0.77 CSNK1A1 (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed