SCHEMBL8537652

SCHEMBL8537652

CCCCOC(=O)NC1CCN(C(=O)c2ccc(-n3ccnc3)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP19A1 P11511 1/20 0.47
LSS P48449 1/20 0.47
KMT2A Q03164 2/20 0.46
HPGD P15428 2/20 0.46
HTT P42858 1/20 0.45
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
MMP1 P03956 2/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534724 0.85 LSS (0.48) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL8538842 0.84 LSS (0.48) CYP3A4LSSKMT2AHTTPDCD1
SCHEMBL9523895 0.83 CYP2C19 (0.60) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL8534755 0.82 LSS (0.46) CYP3A4LSSKMT2AHTTPDCD1
SCHEMBL9589824 0.81 EPHX2 (0.46) CYP3A4LSSKMT2AHTTPDCD1
SCHEMBL8535112 0.81 HTR2A (0.54) CYP3A4LSSKMT2AHTTPDCD1
SCHEMBL9589831 0.79 LSS (0.42) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL8534116 0.78 LSS (0.49) CYP2D6CYP2C19CYP3A4LSSKMT2A
SCHEMBL8539476 0.77 QPCTL (0.44) CYP3A4LSSKMT2AHTTPDCD1
SCHEMBL8539477 0.77 QPCTL (0.44) CYP3A4LSSKMT2AHTTPDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537201-B1 1-[4-(IMIDAZOL-1-YL)BENZOYL]PIPERIDINE DERIVATIVES AS ANTIARRHYTHMIC AGENTS SCHERING AG (DE) 1998-11-18 EP disclosed
US-5189036-A Cardiovascular agents; class III antiarrhythmic agents SCHERING AG (DE) 1993-02-23 US disclosed