SCHEMBL8538265

SCHEMBL8538265

Cc1cc(C)nc(N2CCN(C(=S)C3(C)CCc4c(C)c(O)c(C)c(C)c4O3)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
TSHR P16473 2/20 0.49
USP2 O75604 1/20 0.49
TP53 P04637 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
THPO P40225 1/20 0.49
HIF1A Q16665 1/20 0.49
LCK P06239 1/20 0.49
FYN P06241 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
DRD2 P14416 1/20 0.49
ADRA1D P25100 1/20 0.49
MAPK3 P27361 1/20 0.49
HTR2C P28335 1/20 0.49
MC4R P32245 1/20 0.49
HRH1 P35367 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8543774 0.86 CYP3A4 (0.67) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8543923 0.86 TTPA (0.42) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8543465 0.81 CYP3A4 (0.45) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8544837 0.79 CYP3A4 (0.52) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8540971 0.77 CYP3A4 (0.47) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8539212 0.77 CYP3A4 (0.47) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL9266621 0.76 CYP3A4 (0.46) CYP3A4TSHRCYP2C9LMNAPTGS1
SCHEMBL9256806 0.75 PTGS1 (0.49) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9756674 0.74 CYP3A4 (0.67) CYP3A4TSHRUSP2TP53CYP2C9
SCHEMBL8538881 0.73 PTGS1 (0.49) CYP3A4TSHRPTGS1PTGS2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587499-B1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR (FR) 1998-04-29 EP disclosed
US-5395834-A Antiarthritic agents or cardiovascular disorders ADIR ET COMPAGNIE (FR) 1995-03-07 US disclosed
US-5393775-A Administering a (2-chromanyl)alkylcarboxylic acid for disorders connected with peroxidation processes ADIR ET COMPAGNIE (FR) 1995-02-28 US disclosed
EP-0587499-A1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR ET COMPAGNIE (FR) 1994-03-16 EP disclosed