SCHEMBL8538368

SCHEMBL8538368

CCN(c1ccccc1)c1nc(N2CCOCC2)nc(-n2ccnc2)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 13/20 0.64
NPSR1 Q6W5P4 7/20 0.64
LMNA P02545 6/20 0.64
HTT P42858 6/20 0.64
MAPT P10636 5/20 0.64
TP53 P04637 3/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
HSD17B10 Q99714 1/20 0.64
USP2 O75604 1/20 0.61
ALOX15 P16050 1/20 0.61
MAPK1 P28482 6/20 0.56
KDM4E B2RXH2 1/20 0.56
ATM Q13315 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
L3MBTL1 Q9Y468 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8535479 0.91 TSHR (0.58) TSHRNPSR1LMNAHTTMAPT
SCHEMBL11900640 0.89 TSHR (0.80) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8539849 0.87 TSHR (0.74) TSHRNPSR1LMNAHTTMAPT
SCHEMBL1444931 0.87 TSHR (0.81) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8538515 0.80 TSHR (0.56) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8533688 0.79 LMNA (0.57) TSHRNPSR1LMNAHTTMAPT
SCHEMBL3278610 0.79 LMNA (0.57) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8539843 0.77 TSHR (0.77) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8538506 0.77 TSHR (0.65) TSHRNPSR1LMNAHTTMAPT
SCHEMBL8538662 0.77 TSHR (0.65) TSHRNPSR1LMNAHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0629622-B1 S-TRIAZINE DERIVATIVE AND REMEDY FOR ESTROGEN-DEPENDENT DISEASES CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KK (JP) 1998-11-11 EP disclosed
US-5489591-A INHIBITORS OF AROMATASE; TREATING ENDOMETRIOSIS, BREAST CANCER CYSTIC OVARIES ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 1996-02-06 US disclosed
EP-0629622-A1 s-TRIAZINE DERIVATIVE AND REMEDY FOR ESTROGEN-DEPENDENT DISEASES CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1994-12-21 EP disclosed