SCHEMBL8538571

SCHEMBL8538571

CSC(C)(C)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
TRPV1 Q8NER1 2/20 0.47
SRD5A2 P31213 2/20 0.47
NR4A1 P22736 1/20 0.46
NR4A2 P43354 1/20 0.46
NR4A3 Q92570 1/20 0.46
GSK3B P49841 2/20 0.46
PTPN1 P18031 2/20 0.46
BACE1 P56817 1/20 0.43
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
MMP1 P03956 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7609999 0.83 CES2 (0.55) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL7798781 0.80 CES2 (0.61) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL8235165 0.80 CES2 (0.61) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL7806283 0.79 CES2 (0.59) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL8821889 0.76 CES1 (0.50) CES2CES1MEN1HPGDTSHR
SCHEMBL23172558 0.76 CES2 (0.67) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL1078685 0.76 CES1 (0.67) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL26054729 0.76 CES2 (0.55) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL21387720 0.75 CES2 (0.59) CES2CES1TRPV1SRD5A2NR4A1
SCHEMBL29137235 0.74 CES2 (0.64) CES2CES1TRPV1SRD5A2NR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0435081-B1 Triazole derivatives SS PHARMACEUTICAL CO (JP) 1998-08-12 EP disclosed
US-5147886-A Skin disorders; urogenital,respiratory systems SS PHARMACEUTICAL CO., LTD. (JP) 1992-09-15 US disclosed
EP-0435081-A2 Triazole derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1991-07-03 EP disclosed