SCHEMBL8539162

SCHEMBL8539162

c1ccc(CCCN2CCCC(CCn3ccnc3)C2)cc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.49
SLC6A4 P31645 1/20 0.49
SLC6A3 Q01959 1/20 0.49
CHRNB4 P30926 6/20 0.48
CHRNA3 P32297 6/20 0.48
CHRNB2 P17787 6/20 0.48
CHRNA4 P43681 6/20 0.48
KDM4E B2RXH2 2/20 0.46
KMT2A Q03164 1/20 0.46
CCR2 P41597 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8699420 0.94 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL8539478 0.90 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL8538300 0.86 GRIN2B (0.54)
Hydrochloric Acid SCHEMBL8546852 0.85 GRIN2B (0.53)
SCHEMBL9261150 0.85 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL8545375 0.83 SIGMAR1 (0.59) KMT2A
SCHEMBL9037944 0.82 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL8545836 0.81 HRH3 (0.53)
SCHEMBL8543269 0.81 SIGMAR1 (0.47) KMT2A
SCHEMBL8696473 0.79 SIGMAR1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed