SCHEMBL8539251

SCHEMBL8539251

CSCc1cccnc1-c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.40
MTOR P42345 1/20 0.40
ADK P55263 1/20 0.40
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TAAR1 Q96RJ0 2/20 0.36
HTR1A P08908 1/20 0.36
ADORA2A P29274 3/20 0.35
ADORA1 P30542 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CASP6 P55212 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
IDO1 P14902 1/20 0.32
ADRA2A P08913 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539418 0.81 NISCH (0.42) NISCHMTORADKALDH1A1MEN1
SCHEMBL8537087 0.79 CSNK1A1 (0.45) NISCHMTORADKALDH1A1MEN1
SCHEMBL8541358 0.76 NISCH (0.43) NISCHMTORADKALDH1A1MEN1
SCHEMBL11151750 0.75 CYP1A2 (0.44) NISCHMTORADKTAAR1HTR1A
SCHEMBL29152388 0.73 NISCH (0.48) NISCHMTORADKALDH1A1MEN1
SCHEMBL8536464 0.72 TAAR1 (0.45) NISCHMTORADKALDH1A1MEN1
SCHEMBL8540790 0.71 NISCH (0.37) NISCHMTORADKALDH1A1MEN1
SCHEMBL7537761 0.71 CSNK1A1 (0.49) NISCHMTORADKALDH1A1MEN1
SCHEMBL8537581 0.70 CYP1A2 (0.37) ALDH1A1MEN1KMT2ATAAR1HTR1A
SCHEMBL8535625 0.70 NISCH (0.49) NISCHMTORADKALDH1A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed