SCHEMBL8535625

SCHEMBL8535625

CSCc1cc(-c2ccccc2)ccc1-c1ncc[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.49
MTOR P42345 1/20 0.49
ADK P55263 1/20 0.49
CYP1A2 P05177 2/20 0.37
CSNK1A1 P48729 1/20 0.37
TYRO3 Q06418 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ADORA3 P0DMS8 3/20 0.36
ADORA2A P29274 3/20 0.36
ADORA1 P30542 3/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537087 0.83 CSNK1A1 (0.45) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8540949 0.82 NISCH (0.46) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8540790 0.80 NISCH (0.37) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8536816 0.79 JAK2 (0.47) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8540597 0.79 CSNK1A1 (0.36) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8540730 0.79 MC4R (0.46) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8541400 0.79 MC4R (0.37) NISCHMTORADKCYP1A2CSNK1A1
SCHEMBL8538130 0.79 MAOB (0.43) CYP3A4KDM4E
SCHEMBL8539649 0.77 NOS3 (0.47) NISCHCYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL8539601 0.76 CYP19A1 (0.41) NISCHMTORADKCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed