SCHEMBL8540790

SCHEMBL8540790

CSCc1ccc(-c2ncc[nH]2)c(CSC)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.37
MTOR P42345 1/20 0.35
ADK P55263 1/20 0.35
CSNK1A1 P48729 1/20 0.34
TYRO3 Q06418 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CASP6 P55212 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
MC4R P32245 2/20 0.33
SMPD3 Q9NY59 1/20 0.32
ALDH1A1 P00352 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8541205 0.90 NISCH (0.36) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8536816 0.84 JAK2 (0.47) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8540597 0.84 CSNK1A1 (0.36) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8541400 0.84 MC4R (0.37) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8540730 0.84 MC4R (0.46) NISCHMTORADKCSNK1A1TYRO3
Water SCHEMBL8537122 0.83 CSNK1A1 (0.31) NISCHCSNK1A1TYRO3DYRK1BCASP6
SCHEMBL8537087 0.81 CSNK1A1 (0.45) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8539649 0.81 NOS3 (0.47) NISCHCYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL8535625 0.80 NISCH (0.49) NISCHMTORADKCSNK1A1TYRO3
SCHEMBL8539601 0.80 CYP19A1 (0.41) NISCHMTORADKCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed