SCHEMBL8539874

SCHEMBL8539874

CCOC(=O)c1cn(C2CC2F)c2c(F)c(F)c(F)c(F)c2c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.62
HTT P42858 2/20 0.54
TSHR P16473 2/20 0.48
CASP1 P29466 1/20 0.48
ADRB2 P07550 1/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 1/20 0.39
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
HSD17B10 Q99714 3/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
TP53 P04637 1/20 0.38
RECQL P46063 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4672032 1.00 STAT3 (0.62) STAT3HTTTSHRCASP1ADRB2
SCHEMBL9096244 1.00 STAT3 (0.62) STAT3HTTTSHRCASP1ADRB2
SCHEMBL7997863 0.93 STAT3 (0.54) STAT3HTTTSHRCASP1ADRB2
SCHEMBL8744098 0.93 STAT3 (0.54) STAT3HTTTSHRCASP1ADRB2
SCHEMBL13483600 0.91 STAT3 (0.52) STAT3HTTTSHRCASP1ADRB2
SCHEMBL13483601 0.88 STAT3 (0.48) STAT3HTTTSHRCASP1ADRB2
SCHEMBL1345146 0.86 STAT3 (0.65) STAT3HTTTSHRCASP1ADRB2
SCHEMBL10365215 0.84 STAT3 (0.55) STAT3HTTADRB2KDM4EALDH1A1
SCHEMBL4671582 0.84 STAT3 (0.46) STAT3HTTTSHRCASP1ADRB2
SCHEMBL8537622 0.84 STAT3 (0.45) STAT3HTTTSHRCASP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545642-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-08-13 US claimed
US-5849757-A Pyridonecarboxylic acid derivatives substituted by a bicyclic amino group as antibacterials DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-12-15 US disclosed
US-5545642-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-08-13 US disclosed