SCHEMBL854

SCHEMBL854

Cn1c2c(c3ccccc31)C(=O)NCCC2

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.64
ALB P02768 4/20 0.64
ACHE P22303 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL918 0.92 BRD4 (0.57) BCHEALBACHE
SCHEMBL13345818 0.82 BRD4 (0.51) BCHEALBACHE
SCHEMBL1003026 0.81 MCHR1 (0.52) BCHEALBACHE
SCHEMBL1146660 0.78 HTR2A (0.51)
SCHEMBL7428637 0.78 HTR2A (0.51)
SCHEMBL30223533 0.78 HTR2A (0.51)
SCHEMBL7294032 0.78 BCHE (0.49) BCHEALBACHE
SCHEMBL625913 0.75 HTR6 (0.61) BCHEALBACHE
SCHEMBL984 0.74 HTR2A (0.54)
SCHEMBL3558226 0.73 PTPN1 (0.54) BCHEALBACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360800-A Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives GLAXO GROUP LIMITED (GB) 1994-11-01 US disclosed
EP-0306323-A2 Lactam derivatives GLAXO GROUP LIMITED (GB) 1989-03-08 EP disclosed