SCHEMBL8540459

SCHEMBL8540459

CO[C@H](C(=O)N1CCC[C@@H]1c1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.56
ADAM17 P78536 4/20 0.47
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
RAB9A P51151 1/20 0.45
EPHX2 P34913 2/20 0.44
HSD11B1 P28845 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNA4 P43681 1/20 0.44
SCD5 Q86SK9 3/20 0.44
SCD O00767 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540457 1.00 RIPK1 (0.56) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL8546239 0.96 RIPK1 (0.51) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL8540511 0.96 RIPK1 (0.51) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL8540509 0.96 RIPK1 (0.51) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL8545905 0.95 RIPK1 (0.50) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL8539202 0.95 RIPK1 (0.50) RIPK1ADAM17HSP90AA1HSP90AB1RAB9A
SCHEMBL6439008 0.83 ALDH1A1 (0.53) HSD17B10
SCHEMBL6435766 0.83 ALDH1A1 (0.53) HSD17B10
SCHEMBL6435771 0.83 ALDH1A1 (0.53) HSD17B10
SCHEMBL6436519 0.83 ALDH1A1 (0.53) HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705259-B1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-02-25 EP disclosed
EP-0705259-A1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-10 EP disclosed
WO-1995000508-A1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-01-05 WO disclosed