SCHEMBL8540496

SCHEMBL8540496

OCCc1ccc(Cl)cc1-c1ncc[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.39
CASP6 P55212 1/20 0.38
IDO1 P14902 1/20 0.37
CSNK1A1 P48729 1/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
PIM1 P11309 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CYP19A1 P11511 1/20 0.35
FPR2 P25090 1/20 0.34
JAK2 O60674 2/20 0.34
JAK1 P23458 2/20 0.34
MTOR P42345 1/20 0.34
ADK P55263 1/20 0.34
NISCH Q9Y2I1 1/20 0.34
GRK2 P25098 1/20 0.33
ABL1 P00519 1/20 0.33
GSK3B P49841 1/20 0.33
TYK2 P29597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612212 0.90 MC4R (0.37) MC4RCASP6IDO1CSNK1A1TYRO3
SCHEMBL31429694 0.79 IDO1 (0.51) CASP6IDO1CSNK1A1TYRO3DYRK1B
SCHEMBL6951802 0.78 CSNK1A1 (0.50) MC4RCASP6IDO1CSNK1A1TYRO3
SCHEMBL31429733 0.78 IDO1 (0.58) IDO1CSNK1A1TYRO3DYRK1BPIM1
SCHEMBL29084865 0.78 IDO1 (0.58) IDO1CSNK1A1TYRO3DYRK1BPIM1
SCHEMBL8542466 0.76 ALDH1A1 (0.49) IDO1CSNK1A1TYRO3DYRK1BNPC1
SCHEMBL3631532 0.74 RAB9A (0.50) CSNK1A1TYRO3DYRK1BNPC1RAB9A
SCHEMBL8537019 0.73 IDO1 (0.57) IDO1CSNK1A1TYRO3DYRK1BNPC1
SCHEMBL8558526 0.73 NPC1 (0.40) IDO1CSNK1A1TYRO3DYRK1BPIM1
SCHEMBL8539541 0.73 CYP1A2 (0.43) MC4RCASP6IDO1CSNK1A1TYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed